| The direct acyl-alkylation of arynes UK Tambar, BM Stoltz Journal of the American Chemical Society 127 (15), 5340-5341, 2005 | 365 | 2005 |
| Allosteric inhibition of hypoxia inducible factor-2 with small molecules TH Scheuermann, Q Li, HW Ma, J Key, L Zhang, R Chen, JA Garcia, ... Nature chemical biology 9 (4), 271-276, 2013 | 311 | 2013 |
| Pd-catalyzed enantioselective aerobic oxidation of secondary alcohols: applications to the total synthesis of alkaloids S Krishnan, JT Bagdanoff, DC Ebner, YK Ramtohul, UK Tambar, ... Journal of the American Chemical Society 130 (41), 13745-13754, 2008 | 169 | 2008 |
| A convergent and enantioselective synthesis of (+)-amurensinine via selective C− H and C− C bond insertion reactions UK Tambar, DC Ebner, BM Stoltz Journal of the American Chemical Society 128 (36), 11752-11753, 2006 | 166 | 2006 |
| Development of inhibitors of the PAS-B domain of the HIF-2α transcription factor JL Rogers, L Bayeh, TH Scheuermann, J Longgood, J Key, J Naidoo, ... Journal of medicinal chemistry 56 (4), 1739-1747, 2013 | 138 | 2013 |
| Total synthesis of (±)-Trigonoliimine C via oxidative rearrangement of an unsymmetrical bis-tryptamine X Qi, H Bao, UK Tambar Journal of the American Chemical Society 133 (26), 10050-10053, 2011 | 114 | 2011 |
| Structure-guided development of specific pyruvate dehydrogenase kinase inhibitors targeting the ATP-binding pocket SC Tso, X Qi, WJ Gui, CY Wu, JL Chuang, I Wernstedt-Asterholm, ... Journal of Biological Chemistry 289 (7), 4432-4443, 2014 | 96 | 2014 |
| Catalytic enantioselective allylic amination of unactivated terminal olefins via an ene reaction/[2, 3]-rearrangement H Bao, UK Tambar Journal of the American Chemical Society 134 (45), 18495-18498, 2012 | 91 | 2012 |
| Brønsted acid catalyzed enantioselective indole aza-Claisen rearrangement mediated by an arene CH–O interaction P Maity, RP Pemberton, DJ Tantillo, UK Tambar Journal of the American Chemical Society 135 (44), 16380-16383, 2013 | 89 | 2013 |
| Catalytic allylic oxidation of internal alkenes to a multifunctional chiral building block L Bayeh, PQ Le, UK Tambar Nature 547 (7662), 196-200, 2017 | 88 | 2017 |
| Benzothiophene carboxylate derivatives as novel allosteric inhibitors of branched-chain α-ketoacid dehydrogenase kinase SC Tso, WJ Gui, CY Wu, JL Chuang, X Qi, KJ Skvorak, K Dorko, ... Journal of Biological Chemistry 289 (30), 20583-20593, 2014 | 87 | 2014 |
| Tandem catalytic allylic amination and [2, 3]-Stevens rearrangement of tertiary amines A Soheili, UK Tambar Journal of the American Chemical Society 133 (33), 12956-12959, 2011 | 75 | 2011 |
| Structure-based design and mechanisms of allosteric inhibitors for mitochondrial branched-chain α-ketoacid dehydrogenase kinase SC Tso, X Qi, WJ Gui, JL Chuang, LK Morlock, AL Wallace, K Ahmed, ... Proceedings of the National Academy of Sciences 110 (24), 9728-9733, 2013 | 73 | 2013 |
| Isoform-selective and stereoselective inhibition of hypoxia inducible factor-2 TH Scheuermann, D Stroud, CE Sleet, L Bayeh, C Shokri, H Wang, ... Journal of Medicinal Chemistry 58 (15), 5930-5941, 2015 | 72 | 2015 |
| Ligand-controlled regiodivergence in the copper-catalyzed [2, 3]-and [1, 2]-rearrangements of iodonium ylides B Xu, UK Tambar Journal of the American Chemical Society 138 (37), 12073-12076, 2016 | 63 | 2016 |
| Lactate production is a prioritized feature of adipocyte metabolism JR Krycer, LE Quek, D Francis, DJ Fazakerley, SD Elkington, ... Journal of Biological Chemistry 295 (1), 83-98, 2020 | 60 | 2020 |
| Catalytic Enantioselective [2,3]-Rearrangements of Amine N-Oxides H Bao, X Qi, UK Tambar Journal of the American Chemical Society 133 (5), 1206-1208, 2011 | 60 | 2011 |
| Remote Allylation of Unactivated C(sp3)–H Bonds Triggered by Photogenerated Amidyl Radicals B Xu, UK Tambar ACS catalysis 9 (5), 4627-4631, 2019 | 58 | 2019 |
| A new paradigm for GERD pathogenesis. Not acid injury, but cytokine-mediated inflammation driven by HIF-2α: a potential role for targeting HIF-2α to prevent and treat reflux … RF Souza, L Bayeh, SJ Spechler, UK Tambar, RK Bruick Current opinion in pharmacology 37, 93-99, 2017 | 58 | 2017 |
| Copper‐Catalyzed Enantio‐, Diastereo‐, and Regioselective [2, 3]‐Rearrangements of Iodonium Ylides B Xu, UK Tambar Angewandte Chemie International Edition 56 (33), 9868-9871, 2017 | 53 | 2017 |
Brian StoltzProfessor of Chemistry, California Institute of TechnologyVerified email at caltech.edu
