Reliability of logP predictions based on calculated molecular descriptors: a critical review D Eros, I Kovesdi, L Orfi, K Takacs-Novak, G Acsády, G Kéri Current medicinal chemistry 9 (20), 1819-1829, 2002 | 135 | 2002 |
A novel drug discovery concept for tuberculosis: inhibition of bacterial and host cell signalling R Székely, F Wáczek, I Szabadkai, G Németh, B Hegymegi-Barakonyi, ... Immunology letters 116 (2), 225-231, 2008 | 102 | 2008 |
Signal transduction therapy with rationally designed kinase inhibitors G Keri, L Orfi, D Eros, B Hegymegi-Barakonyi, C Szantai-Kis, Z Horvath, ... Current Signal Transduction Therapy 1 (1), 67-95, 2006 | 67 | 2006 |
Comparison of predictive ability of water solubility QSPR models generated by MLR, PLS and ANN methods D Eros, G Keri, I Kovesdi, C Szantai-Kis, G Meszaros, L Orfi Mini Reviews in Medicinal Chemistry 4 (2), 167-177, 2004 | 59 | 2004 |
Binding mode analysis and enrichment studies on homology models of the human histamine H4 receptor R Kiss, B Noszál, Á Rácz, A Falus, D Erős, GM Keserű European journal of medicinal chemistry 43 (5), 1059-1070, 2008 | 56 | 2008 |
Signalling inhibitors against Mycobacterium tuberculosis-early days of a new therapeutic concept in tuberculosis B Hegymegi-Barakonyi, R Szekely, Z Varga, R Kiss, G Borbely, G Nemeth, ... Current medicinal chemistry 15 (26), 2760-2770, 2008 | 47 | 2008 |
Drug discovery in the kinase inhibitory field using the nested chemical library™ technology G Kéri, Z Székelyhidi, P Bánhegyi, Z Varga, B Hegymegi-Barakonyi, ... Assay and drug development technologies 3 (5), 543-551, 2005 | 43 | 2005 |
Relationship between lipophilicity and antitumor activity of molecule library of Mannich ketones determined by high-performance liquid chromatography, clogP calculation and … F Hollósy, T Lóránd, L Örfi, D Erös, G Kéri, M Idei Journal of Chromatography B 768 (2), 361-368, 2002 | 42 | 2002 |
Comparison of measured and calculated lipophilicity of substituted aurones and related compounds B Hallgas, T Patonay, A Kiss-Szikszai, Z Dobos, F Hollósy, D Erős, L Őrfi, ... Journal of Chromatography B 801 (2), 229-235, 2004 | 39 | 2004 |
Tyrosine kinase inhibitors-small molecular weight compounds inhibiting EGFR. B Hegymegi-Barakonyi, D Eros, C Szantai-Kis, N Breza, P Bánhegyi, ... Current Opinion in Molecular Therapeutics 11 (3), 308-321, 2009 | 29 | 2009 |
Characterization of lipophilicity and antiproliferative activity of E-2-arylmethylene-1-tetralones and their heteroanalogues B Hallgas, Z Dobos, E Ősz, F Hollósy, RE Schwab, EZ Szabó, D Erős, ... Journal of Chromatography B 819 (2), 283-291, 2005 | 28 | 2005 |
Evaluation of lipophilicity and antitumour activity of parallel carboxamide libraries F Hollósy, J Seprödi, L Örfi, D Erös, G Kéri, M Idei Journal of Chromatography B 780 (2), 355-363, 2002 | 27 | 2002 |
Biological activity and structure of antitumor compounds from Plantago media L M Kunvari, C Paska, M Laszlo, L Orfi, I Kövesdi, D Eros, G Bökönyi, G Keri, ... Acta Pharmaceutica Hungarica 69 (5), 232-239, 1999 | 25 | 1999 |
Regulation of influenza A virus mRNA splicing by CLK1 A Artarini, M Meyer, YJ Shin, K Huber, N Hilz, F Bracher, D Eros, L Orfi, ... Antiviral research 168, 187-196, 2019 | 24 | 2019 |
Structure-Activity Relationships of PDE5 Inhibitors (Supporting Material) D Eros, C Szantai-Kis, R Kiss, G Keri, B Hegymegi-Barakonyi, I Kovesdi, ... Current medicinal chemistry 15 (16), 1570-1585, 2008 | 24 | 2008 |
Prediction oriented QSAR modelling of EGFR inhibition C Szantai-Kis, I Kovesdi, D Eros, P Bánhegyi, A Ullrich, G Kéri, L Orfi Current Medicinal Chemistry 13 (3), 277-287, 2006 | 23 | 2006 |
Targeted drug combination therapy design based on driver genes L Zsákai, A Sipos, J Dobos, D Erős, C Szántai-Kis, P Bánhegyi, J Pató, ... Oncotarget 10 (51), 5255, 2019 | 20 | 2019 |
Determination of the basicity of Mannich ketones by capillary electrophoresis Z Dobos, T Lóránd, F Hollósy, B Hallgas, D Erős, GY Mészáros, GY Kéri, ... Journal of Chromatography B 799 (1), 179-183, 2004 | 14 | 2004 |
Evaluation of hydrophobicity and antitumor activity of a molecule library of mannich ketones of cycloalkanones F Hollosy, T Lorand, L Őrfi, D Erős, G Kéri, M Idei Journal of liquid chromatography & related technologies 25 (7), 1129-1143, 2002 | 8 | 2002 |
MIF tautomerase inhibitor potency of α, β-unsaturated cyclic ketones J Garai, V Molnár, D Erős, L Őrfi, T Lóránd International immunopharmacology 7 (13), 1741-1746, 2007 | 7 | 2007 |