2-[N-Acylamino(C1−C3)alkyl]indoles as MT1 Melatonin Receptor Partial Agonists, Antagonists, and Putative Inverse Agonists G Spadoni, C Balsamini, A Bedini, G Diamantini, B Di Giacomo, A Tontini, ... Journal of medicinal chemistry 41 (19), 3624-3634, 1998 | 128 | 1998 |
Melatonin receptor ligands: Synthesis of new melatonin derivatives and comprehensive comparative molecular field analysis (CoMFA) study M Mor, S Rivara, C Silva, F Bordi, PV Plazzi, G Spadoni, G Diamantini, ... Journal of medicinal chemistry 41 (20), 3831-3844, 1998 | 100 | 1998 |
Conformationally restrained melatonin analogues: synthesis, binding affinity for the melatonin receptor, evaluation of the biological activity, and molecular modeling study G Spadoni, C Balsamini, G Diamantini, B Di Giacomo, G Tarzia, M Mor, ... Journal of medicinal chemistry 40 (13), 1990-2002, 1997 | 91 | 1997 |
Switchable reactivity of acylated α, β-dehydroamino ester in the Friedel− Crafts alkylation of indoles by changing the Lewis acid E Angelini, C Balsamini, F Bartoccini, S Lucarini, G Piersanti The Journal of Organic Chemistry 73 (14), 5654-5657, 2008 | 83 | 2008 |
2-N-Acylaminoalkylindoles: Design and Quantitative Structure−Activity Relationship Studies Leading to MT2-Selective Melatonin Antagonists G Spadoni, C Balsamini, G Diamantini, A Tontini, G Tarzia, M Mor, ... Journal of medicinal chemistry 44 (18), 2900-2912, 2001 | 69 | 2001 |
A new melatonin receptor ligand with mt1‐agonist and MT2‐antagonist properties R Nonno, V Lucini, G Spadoni, M Pannacci, A Croce, D Esposti, ... Journal of pineal research 29 (4), 234-240, 2000 | 40 | 2000 |
Structural requirements for inhibitors of poly (ADP-ribose) polymerase P Sestili, G Spadoni, C Balsamini, I Scovassi, F Cattabeni, E Duranti, ... Journal of cancer research and clinical oncology 116, 615-622, 1990 | 34 | 1990 |
Stereospecific Synthesis of N-(Diphenylmethylene)-α, β-didehydroamino Acid Methyl Esters from β-Hydroxy-α-amino Acids C Balsamini, E Duranti, L Mariani, A Salvatori, G Spadoni Synthesis 1990 (09), 779-781, 1990 | 28 | 1990 |
Alkyl 2-(diphenylmethyleneamino) acrylates in the synthesis of α-amino acids G Tarzia, C Balsamini, G Spadoni, E Duranti Synthesis 1988 (07), 514-517, 1988 | 24 | 1988 |
(E)-3-(2-(N-phenylcarbamoyl) vinyl) pyrrole-2-carboxylic acid derivatives. A novel class of glycine site antagonists C Balsamini, A Bedini, G Diamantini, G Spadoni, A Tontini, G Tarzia, ... Journal of medicinal chemistry 41 (6), 808-820, 1998 | 23 | 1998 |
Reactions of 3-carbomethoxy-2-aza-1, 3-butadiene derivatives with dienophiles C Balsamini, A Bedini, R Galarini, G Spadoni, G Tarzia, M Hamdan Tetrahedron 50 (43), 12375-12394, 1994 | 23 | 1994 |
Synthetic approaches to nitro-substituted isoxazoles DA Vasilenko, KN Sedenkova, TS Kuznetsova, EB Averina Synthesis 51 (07), 1516-1528, 2019 | 22 | 2019 |
N-Acyl-5-and-2, 5-substituted tryptamines: synthesis, activity and affinity for human mt1 and MT2 melatonin receptors G Spadoni, C Balsamini, A Bedini, A Carey, G Diamantini, B DI GIACOMO, ... Medicinal Chemistry Research 8, 487-498, 1998 | 21 | 1998 |
Reaction of secondary acetylenic bromides with sodium nitrite: synthesis of 3, 5-alkyl (aryl)-4-nitroisoxazoles E Duranti, C Balsamini, G Spadoni, L Staccioli The Journal of Organic Chemistry 53 (12), 2870-2872, 1988 | 20 | 1988 |
Analogues of benzamide containing a sulfur atom as poly (ADP-ribose) transferase inhibitors. O Cantoni, P Sestili, G Spadoni, C Balsamini, L Cucchiarini, F Cattabeni Biochemistry international 15 (2), 329-337, 1987 | 20 | 1987 |
Short synthesis of tryptophane and β‐carboline derivatives by reaction of indoles with N‐(diphenylmethylene)‐α,β‐didehydroamino acid esters G Spadoni, C Balsamini, A Bedini, E Duranti, A Tontini Journal of heterocyclic chemistry 29 (2), 305-309, 1992 | 19 | 1992 |
Synthesis of 1-(isoxazol-3-yl) triazene derivatives. Antimetastatic activity of 3, 3-dimethyl-1-(5-methylisoxazol-3-yl) triazene A Tontini, G Diamantini, C Balsamini, G Tarzia, L Perissin, V Rapozzi European journal of medicinal chemistry 31 (9), 735-740, 1996 | 18 | 1996 |
4,5‐Dihydroisoxazole and 4,5‐dihydro‐1,2,4‐oxadiazole derivatives from cycloaddition reactions of nitrile oxides to alkyl N‐(diphenylmethylene)‐α,β … C Balsamini, G Spadoni, A Bedini, G Tarzia, M Lanfranchi, MA Pellinghelli Journal of heterocyclic chemistry 29 (6), 1593-1598, 1992 | 15 | 1992 |
Positive‐ion mass spectra and collision‐induced dissociation of some 2, 3‐didehydro amino acids M Hamdan, G Tarzia, C Balsamini, G Spadoni, O Curcuruto, P Traldi Organic mass spectrometry 25 (10), 540-549, 1990 | 15 | 1990 |
A New Synthetic Route to 2,2′-Biimidazole E Duranti, B Cesarino Synthesis 1974 (1), 1974 | 14 | 1974 |